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ML334

Glpbio
Catalog No:GC38819-10mM (in 1mL DMSO) CAS No.:1432500-66-7 MDLNo: Brand:Glpbio purity: 特性: Purpose:ML334 (LH601A) 是一种有效的,细胞可渗透的 NRF2 激活剂,通过抑制 Keap1-NRF2 蛋白质相互作用来发挥作用。ML334 以 Kd 值为 1μM 来结合 Keap1 Kelch 域。ML334 刺激 NRF2 表达和核易位并诱导抗氧化反应元件 (ARE) 活性。DMSO: 44.65 mg/mL (100.00 mM); Ethanol: 44.65 mg/mL (100.00 mM)
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